Kinetic data for "OXA%"
Number of results: 267
| # |
Protein Name |
Antibiotic |
kcat (s-1) |
Km (µM) |
kcat/KM |
| 1 |
OXA-11 |
Benzylpenicillin |
|
42 |
|
| 2 |
OXA-11 |
Cefotaxime |
|
8.5 |
|
| 3 |
OXA-11 |
Ampicillin |
|
35 |
|
| 4 |
OXA-11 |
Cephalothin |
|
12 |
|
| 5 |
OXA-11 |
Oxacillin |
|
Nonlinear |
|
| 6 |
OXA-11 |
Ceftazidime |
|
1.1 |
|
| 7 |
OXA-11 |
Cephaloridine |
|
3.6 |
|
| 8 |
OXA-114 |
Cefoxitin |
<0.01 |
|
|
| 9 |
OXA-114 |
Cephalothin |
0.5 |
15 |
0.03 |
| 10 |
OXA-114 |
Imipenem |
>0.1 |
>2100 |
0 |
| 11 |
OXA-114 |
Oxacillin |
<0.01 |
|
|
| 12 |
OXA-114 |
Ceftazidime |
<0.01 |
|
|
| 13 |
OXA-114 |
Piperacillin |
0.5 |
1 |
0.1 |
| 14 |
OXA-114 |
Ticarcillin |
0.1 |
40 |
0 |
| 15 |
OXA-114 |
Benzylpenicillin |
0.1 |
10 |
0.01 |
| 16 |
OXA-114 |
Cefotaxime |
<0.01 |
|
|
| 17 |
OXA-143 |
Cephalothin |
0.2 |
220 |
0 |
| 18 |
OXA-143 |
Ampicillin |
7 |
700 |
0.01 |
| 19 |
OXA-143 |
Aztreonam |
<0.01 |
|
|
| 20 |
OXA-143 |
Imipenem |
|
0.05 |
5 |
| 21 |
OXA-143 |
Oxacillin |
1.2 |
450 |
0 |
| 22 |
OXA-143 |
Ceftazidime |
<0.01 |
|
|
| 23 |
OXA-143 |
Cefepime |
<0.01 |
|
|
| 24 |
OXA-143 |
Piperacillin |
1 |
40 |
0.03 |
| 25 |
OXA-143 |
Ticarcillin |
1 |
370 |
0 |
| 26 |
OXA-143 |
Meropenem |
0.3 |
100 |
0 |
| 27 |
OXA-143 |
Benzylpenicillin |
5 |
80 |
0.06 |
| 28 |
OXA-143 |
Cefotaxime |
<0.01 |
|
|
| 29 |
OXA-143 |
Cefoxitin |
<0.01 |
|
|
| 30 |
OXA-143 |
Ertapenem |
0.01 |
|
|
| 31 |
OXA-145 |
Imipenem |
<0.01 |
NA |
NA |
| 32 |
OXA-145 |
Oxacillin |
<0.1 |
NA |
NA |
| 33 |
OXA-145 |
Ceftazidime |
0.4 |
18 |
0.02 |
| 34 |
OXA-145 |
Cefepime |
<0.05 |
NA |
NA |
| 35 |
OXA-145 |
Piperacillin |
<0.02 |
NA |
NA |
| 36 |
OXA-145 |
Ticarcillin |
<0.1 |
NA |
NA |
| 37 |
OXA-145 |
Nitrocefine |
1.2 |
38 |
0.03 |
| 38 |
OXA-145 |
Cefotaxime |
<0.2 |
NA |
NA |
| 39 |
OXA-145 |
Penicillin G |
<0.05 |
NA |
NA |
| 40 |
OXA-145 |
Cephaloridine |
1.4 |
100 |
0.01 |
| 41 |
OXA-145 |
Cefoxitin |
<0.1 |
NA |
NA |
| 42 |
OXA-145 |
Cefuroxime |
1 |
70 |
0.02 |
| 43 |
OXA-145 |
Ampicillin |
0.3 |
5 |
52 |
| 44 |
OXA-145 |
Aztreonam |
|
NA |
NA |
| 45 |
OXA-163 |
Cefepime |
2 |
350 |
0.01 |
| 46 |
OXA-163 |
Piperacillin |
8 |
70 |
0.11 |
| 47 |
OXA-163 |
Ticarcillin |
1 |
320 |
0 |
| 48 |
OXA-163 |
Meropenem |
0.07 |
2200 |
0 |
| 49 |
OXA-163 |
Cefotaxime |
30 |
850 |
35 |
| 50 |
OXA-163 |
Benzylpenicillin |
15 |
40 |
0.38 |
| 51 |
OXA-163 |
Ertapenem |
0.01 |
150 |
0 |
| 52 |
OXA-163 |
Ampicillin |
25 |
320 |
0.08 |
| 53 |
OXA-163 |
Aztreonam |
0.5 |
230 |
0 |
| 54 |
OXA-163 |
Cephalothin |
3 |
80 |
0.04 |
| 55 |
OXA-163 |
Imipenem |
0.03 |
530 |
0 |
| 56 |
OXA-163 |
Ceftazidime |
200 |
>2000 |
1 |
| 57 |
OXA-18 |
Ticarcillin |
|
12 |
|
| 58 |
OXA-18 |
Cefotaxime |
|
23 |
|
| 59 |
OXA-18 |
Benzylpenicillin |
|
2.5 |
|
| 60 |
OXA-18 |
Cephaloridine |
|
132 |
|
| 61 |
OXA-18 |
Ampicillin |
|
1.3 |
|
| 62 |
OXA-18 |
Aztreonam |
|
3 |
|
| 63 |
OXA-18 |
Cephalothin |
|
26.5 |
|
| 64 |
OXA-18 |
Ceftazidime |
|
499 |
|
| 65 |
OXA-18 |
Cefepime |
|
64 |
|
| 66 |
OXA-198 |
Meropenem |
0.01 |
0.01 |
1.67 |
| 67 |
OXA-198 |
Benzylpenicillin |
15 |
14 |
1.07 |
| 68 |
OXA-198 |
Ampicillin |
37 |
216 |
0.17 |
| 69 |
OXA-198 |
Cephalothin |
0.19 |
12 |
0.02 |
| 70 |
OXA-198 |
Imipenem |
0.1 |
0.15 |
0.67 |
| 71 |
OXA-198 |
Piperacillin |
2.6 |
35 |
0.07 |
| 72 |
OXA-198 |
Oxacillin |
25 |
30 |
0.83 |
| 73 |
OXA-20 |
Cephaloridine |
20±0.90 |
69±5.00 |
0.3±0.009 |
| 74 |
OXA-20 |
Ampicillin |
80±1.40 |
33±2.20 |
2.4±0.13 |
| 75 |
OXA-20 |
Cephalothin |
13±0.05 |
5±0.20 |
2.6±0.08 |
| 76 |
OXA-20 |
Penicillin G |
26±0.90 |
4.4±1.30 |
5.9±1.70 |
| 77 |
OXA-20 |
Cloxacillin |
70±7 |
329±114 |
0.088±0.005 |
| 78 |
OXA-20 |
Aztreonam |
6±0.50 |
69±12.00 |
0.09±0.009 |
| 79 |
OXA-20 |
Oxacillin |
116±5 |
329±34 |
0.35±0.020 |
| 80 |
OXA-20 |
Ticarcillin |
4±0.45 |
147±34 |
0.03±0.004 |
| 81 |
OXA-22 |
Amoxicillin |
0.1 |
6 |
0.02 |
| 82 |
OXA-22 |
Benzylpenicillin |
0.1 |
<2 |
>0.04 |
| 83 |
OXA-22 |
Cephaloridine |
5.5 |
10 |
0.55 |
| 84 |
OXA-22 |
Cephalothin |
0.9 |
3 |
0.33 |
| 85 |
OXA-22 |
Cloxacillin |
0.7 |
5 |
0.14 |
| 86 |
OXA-22 |
Cefoxitin |
0.05 |
10 |
0 |
| 87 |
OXA-22 |
Ticarcillin |
0.1 |
9 |
0.01 |
| 88 |
OXA-22 |
Cefuroxime |
0.05 |
5 |
0.01 |
| 89 |
OXA-229 |
Cephalothin |
0.2 |
165 |
0 |
| 90 |
OXA-229 |
Meropenem |
<0.01 |
0.03 |
<0.00001 |
| 91 |
OXA-229 |
Ampicillin |
1 |
127 |
0.01 |
| 92 |
OXA-229 |
Ticarcillin |
1.7 |
343 |
0.01 |
| 93 |
OXA-229 |
Imipenem |
0.09 |
30 |
0 |
| 94 |
OXA-229 |
Oxacillin |
4.2 |
1850 |
0 |
| 95 |
OXA-229 |
Piperacillin |
2.2 |
29 |
0.08 |
| 96 |
OXA-229 |
Amoxicillin |
15.2 |
405 |
0.04 |
| 97 |
OXA-229 |
Benzylpenicillin |
11 |
70 |
0.15 |
| 98 |
OXA-235 |
Ampicillin |
0.73±0.015 |
85±21 |
0.01 |
| 99 |
OXA-235 |
Nitrocefine |
65.64±7 |
53±7 |
1.23 |
| 100 |
OXA-235 |
Imipenem |
0.066±0.01 |
0.19±0.043 |
0.34 |
| 101 |
OXA-235 |
Oxacillin |
110±27 |
818±139 |
0.13 |
| 102 |
OXA-235 |
Meropenem |
0.117±0.023 |
0.0159±0.0027 |
7.35 |
| 103 |
OXA-24 |
Cephaloridine |
|
395 |
|
| 104 |
OXA-24 |
Imipenem |
|
20 |
|
| 105 |
OXA-24 |
Meropenem |
|
775 |
|
| 106 |
OXA-24 |
Benzylpenicillin |
|
65 |
|
| 107 |
OXA-25 |
Cefotaxime |
|
35 |
|
| 108 |
OXA-25 |
Imipenem |
|
11 |
|
| 109 |
OXA-25 |
Penicillin G |
|
100 |
|
| 110 |
OXA-25 |
Oxacillin |
|
840 |
|
| 111 |
OXA-25 |
Carbenicillin |
|
300 |
|
| 112 |
OXA-25 |
Cefuroxime |
|
105 |
|
| 113 |
OXA-25 |
Piperacillin |
|
55 |
|
| 114 |
OXA-25 |
Meropenem |
|
12 |
|
| 115 |
OXA-25 |
Cephaloridine |
|
590 |
|
| 116 |
OXA-25 |
Ampicillin |
|
21 |
|
| 117 |
OXA-25 |
Cephalothin |
|
80 |
|
| 118 |
OXA-26 |
Penicillin G |
|
25 |
|
| 119 |
OXA-26 |
Oxacillin |
|
580 |
|
| 120 |
OXA-26 |
Carbenicillin |
|
210 |
|
| 121 |
OXA-26 |
Cefuroxime |
|
7 |
|
| 122 |
OXA-26 |
Piperacillin |
|
10 |
|
| 123 |
OXA-26 |
Meropenem |
|
3 |
|
| 124 |
OXA-26 |
Cephaloridine |
|
640 |
|
| 125 |
OXA-26 |
Ampicillin |
|
15 |
|
| 126 |
OXA-26 |
Cephalothin |
|
90 |
|
| 127 |
OXA-26 |
Imipenem |
|
3 |
|
| 128 |
OXA-27 |
Oxacillin |
|
402 |
|
| 129 |
OXA-27 |
Cefuroxime |
|
2 |
|
| 130 |
OXA-27 |
Piperacillin |
|
10 |
|
| 131 |
OXA-27 |
Meropenem |
|
15 |
|
| 132 |
OXA-27 |
Cephaloridine |
|
3 |
|
| 133 |
OXA-27 |
Ampicillin |
|
3 |
|
| 134 |
OXA-27 |
Cephalothin |
|
260 |
|
| 135 |
OXA-27 |
Imipenem |
|
20 |
|
| 136 |
OXA-27 |
Cefotaxime |
|
0.1 |
|
| 137 |
OXA-27 |
Penicillin G |
|
88 |
|
| 138 |
OXA-29 |
Piperacillin |
31±3 |
39±3 |
0.79 |
| 139 |
OXA-29 |
Carbenicillin |
13±1 |
16±1 |
0.81 |
| 140 |
OXA-29 |
Nitrocefine |
1800±150 |
96±6 |
19 |
| 141 |
OXA-29 |
Cefuroxime |
>0.19 |
>250 |
0 |
| 142 |
OXA-29 |
Aztreonam |
0.21±0.02 |
210±17 |
0 |
| 143 |
OXA-29 |
Ampicillin |
107±10 |
16±1 |
6.7 |
| 144 |
OXA-29 |
Ceftazidime |
>0.24 |
>500 |
0 |
| 145 |
OXA-29 |
Cefotaxime |
0.17±0.01 |
128±11 |
0 |
| 146 |
OXA-29 |
Penicillin G |
27±2 |
41±4 |
0.66 |
| 147 |
OXA-29 |
Oxacillin |
34±3 |
4.4±0.3 |
7.7 |
| 148 |
OXA-31 |
Cloxacillin |
|
2 |
|
| 149 |
OXA-31 |
Cefpirome |
|
120 |
|
| 150 |
OXA-31 |
Cephalothin |
|
45 |
|
| 151 |
OXA-31 |
Cefotaxime |
|
35 |
|
| 152 |
OXA-31 |
Benzylpenicillin |
|
5 |
|
| 153 |
OXA-31 |
Amoxicillin |
|
60 |
|
| 154 |
OXA-31 |
Cefepime |
|
200 |
|
| 155 |
OXA-32 |
Cephalothin |
3 |
60 |
50 |
| 156 |
OXA-32 |
Ticarcillin |
1 |
60 |
15 |
| 157 |
OXA-32 |
Cephaloridine |
3 |
360 |
6 |
| 158 |
OXA-32 |
Benzylpenicillin |
3.5 |
45 |
80 |
| 159 |
OXA-32 |
Ceftazidime |
|
>3000 |
|
| 160 |
OXA-32 |
Amoxicillin |
1.5 |
220 |
70 |
| 161 |
OXA-32 |
Piperacillin |
3 |
155 |
20 |
| 162 |
OXA-32 |
Cloxacillin |
2.5 |
110 |
20 |
| 163 |
OXA-46 |
Cephalothin |
8 |
23 |
0.35 |
| 164 |
OXA-46 |
Aztreonam |
|
>1000 |
|
| 165 |
OXA-46 |
Ampicillin |
6 |
20 |
0.3 |
| 166 |
OXA-46 |
Ceftazidime |
|
>1000 |
|
| 167 |
OXA-46 |
Cefotaxime |
|
>1000 |
|
| 168 |
OXA-46 |
Cefepime |
|
>1000 |
|
| 169 |
OXA-46 |
Penicillin G |
18 |
48 |
0.38 |
| 170 |
OXA-46 |
Oxacillin |
300 |
320 |
0.94 |
| 171 |
OXA-46 |
Carbenicillin |
85 |
730 |
0.12 |
| 172 |
OXA-46 |
Nitrocefine |
20 |
18 |
1.11 |
| 173 |
OXA-46 |
Cefuroxime |
|
>1000 |
|
| 174 |
OXA-48 |
Cephalothin |
3 |
20 |
0.15 |
| 175 |
OXA-48 |
Ampicillin |
340 |
5200 |
0.07 |
| 176 |
OXA-48 |
Cefpirome |
8 |
390 |
0.02 |
| 177 |
OXA-48 |
Meropenem |
0.1 |
200 |
0.01 |
| 178 |
OXA-48 |
Ceftazidime |
4 |
5100 |
0 |
| 179 |
OXA-48 |
Ticarcillin |
45 |
55 |
0.82 |
| 180 |
OXA-48 |
Cephaloridine |
2 |
27 |
0.08 |
| 181 |
OXA-48 |
Cefotaxime |
10 |
190 |
0.06 |
| 182 |
OXA-48 |
Benzylpenicillin |
245 |
40 |
6.1 |
| 183 |
OXA-48 |
Cefepime |
1 |
160 |
0.01 |
| 184 |
OXA-48 |
Oxacillin |
25 |
30 |
0.85 |
| 185 |
OXA-48 |
Imipenem |
2 |
14 |
0.15 |
| 186 |
OXA-48 |
Piperacillin |
75 |
410 |
0.18 |
| 187 |
OXA-54 |
Meropenem |
0.1 |
125 |
0 |
| 188 |
OXA-54 |
Ticarcillin |
30 |
240 |
0 |
| 189 |
OXA-54 |
Cephaloridine |
1 |
45 |
0 |
| 190 |
OXA-54 |
Cefotaxime |
15 |
1600 |
0 |
| 191 |
OXA-54 |
Benzylpenicillin |
120 |
60 |
0 |
| 192 |
OXA-54 |
Cefepime |
1 |
180 |
0 |
| 193 |
OXA-54 |
Oxacillin |
35 |
75 |
0 |
| 194 |
OXA-54 |
Imipenem |
1 |
4 |
0 |
| 195 |
OXA-54 |
Piperacillin |
20 |
240 |
0 |
| 196 |
OXA-54 |
Cephalothin |
3 |
230 |
0 |
| 197 |
OXA-54 |
Ampicillin |
540 |
4300 |
0 |
| 198 |
OXA-54 |
Cefpirome |
4 |
110 |
0 |
| 199 |
OXA-57 |
Oxacillin |
1.23±0.2 |
40.7±6.1 |
0.03 |
| 200 |
OXA-57 |
Piperacillin |
2.11±0.4 |
21.3±3.8 |
0.1 |
| 201 |
OXA-57 |
Penicillin G |
0.40±0.1 |
29.5±5.1 |
0.01 |
| 202 |
OXA-57 |
Cephalothin |
0.28±0.1 |
163±11 |
0 |
| 203 |
OXA-57 |
Cloxacillin |
0.51±0.1 |
28.7±4.2 |
0.02 |
| 204 |
OXA-57 |
Ampicillin |
0.54±0.1 |
71.9±9.6 |
0.01 |
| 205 |
OXA-57 |
Nitrocefine |
63±7.5 |
17.9±2.1 |
3.51 |
| 206 |
OXA-57 |
Cephaloridine |
13±1.9 |
97.9±15 |
0.13 |
| 207 |
OXA-58 |
Benzylpenicillin |
5.5 |
50 |
0.11 |
| 208 |
OXA-58 |
Oxacillin |
1.5 |
70 |
0 |
| 209 |
OXA-58 |
Piperacillin |
2.5 |
50 |
0.05 |
| 210 |
OXA-58 |
Imipenem |
0.1 |
7.5 |
0.01 |
| 211 |
OXA-58 |
Cephalothin |
0.1 |
150 |
0 |
| 212 |
OXA-58 |
Ampicillin |
1 |
130 |
0.01 |
| 213 |
OXA-58 |
Cefpirome |
0.1 |
200 |
0 |
| 214 |
OXA-58 |
Meropenem |
<0.01 |
0.08 |
<0.0015 |
| 215 |
OXA-58 |
Ticarcillin |
1 |
240 |
0 |
| 216 |
OXA-60 |
Ceftazidime |
2 |
1000 |
0 |
| 217 |
OXA-60 |
Piperacillin |
>300 |
>2000 |
<0.150 |
| 218 |
OXA-60 |
Imipenem |
0.5 |
2 |
0.26 |
| 219 |
OXA-60 |
Amoxicillin |
60 |
300 |
0.19 |
| 220 |
OXA-60 |
Cloxacillin |
70 |
1500 |
0.05 |
| 221 |
OXA-60 |
Nitrocefine |
500 |
380 |
1.4 |
| 222 |
OXA-60 |
Ticarcillin |
200 |
400 |
0.52 |
| 223 |
OXA-60 |
Cephaloridine |
>0.5 |
>1000 |
<0.0005 |
| 224 |
OXA-60 |
Benzylpenicillin |
420 |
40 |
11.35 |
| 225 |
OXA-60 |
Oxacillin |
>130 |
>2000 |
<0.065 |
| 226 |
OXA-62 |
Imipenem |
|
13±1.4 |
|
| 227 |
OXA-62 |
Cefoxitin |
|
68±1.4 |
|
| 228 |
OXA-62 |
Ampicillin |
|
160±2.1 |
|
| 229 |
OXA-62 |
Cephaloridine |
|
3200±500 |
|
| 230 |
OXA-62 |
Benzylpenicillin |
|
28±2.3 |
|
| 231 |
OXA-62 |
Meropenem |
|
8.0±2.8 |
|
| 232 |
OXA-62 |
Oxacillin |
|
35±5.5 |
|
| 233 |
OXA-62 |
Piperacillin |
|
13±5.7 |
|
| 234 |
OXA-63 |
Ampicillin |
6.6 |
43 |
0.15 |
| 235 |
OXA-63 |
Benzylpenicillin |
4.9 |
19 |
0.25 |
| 236 |
OXA-63 |
Oxacillin |
113 |
115 |
0.98 |
| 237 |
OXA-63 |
Carbenicillin |
1.1 |
17 |
0.07 |
| 238 |
OXA-63 |
Piperacillin |
2.1 |
33 |
0.06 |